Drug Inventory For Clinical Testing

KYAN has over 100 drugs in inventory to be used for drug sensitivity testing with the Optim.AI™ platform without any lead time. 

If your desired drug is not part of our inventory and it is a drug we can test in our assay, our team can source the drug within weeks.  

Nr.Drug NameDrug ClassificationBiological Target
1AbemaciclibKinase InhibitorCDK4, CDK6
2AcalabrutinibKinase InhibitorBTK (Bruton's Tyrosine Kinase)
3AfatinibKinase InhibitorEGFR (ErbB1), HER2, ErbB4
4AlectinibKinase InhibitorALK (Anaplastic Lymphoma Kinase)
5AlpelisibKinase InhibitorPI3Kα (Phosphatidylinositol 3-kinase)
6AnastrozoleHormonal TherapyAromatase (CYP19A1)
7AvapritinibKinase InhibitorKIT (Exon 17), PDGFRA (Exon 18)
8AzacitidineAntimetabolite (Epigenetic)DNMT (DNA Methyltransferase) / RNA
9BendamustineAlkylating AgentDNA (Cross-linking)
10BinimetinibKinase InhibitorMEK1, MEK2
11BleomycinAntitumor AntibioticDNA (Strand Scission)
12BortezomibProteasome Inhibitor26S Proteasome (Beta-5 subunit)
13CabozantinibKinase InhibitorVEGFR2, MET, RET, AXL
14Capecitabine (5-FU)AntimetaboliteThymidylate Synthase (via 5-FU)
15CapivasertibKinase InhibitorAKT (Protein Kinase B)
16CarboplatinAlkylating AgentDNA (Cross-linking)
17CarfilzomibProteasome Inhibitor20S Proteasome
18CarmustineAlkylating AgentDNA (O6-guanine alkylation)
19CeritinibKinase InhibitorALK
20CetuximabMonoclonal AntibodyEGFR (ErbB1)
21ChlorambucilAlkylating AgentDNA (Cross-linking)
22CisplatinAlkylating AgentDNA (Cross-linking)
23CladribineAntimetaboliteDNA Polymerase / Ribonucleotide Reductase
24ClofarabineAntimetaboliteDNA Polymerase / Ribonucleotide Reductase
25CobimetinibKinase InhibitorMEK1
26CopanlisibKinase InhibitorPI3K (Alpha, Delta isoforms)
27CrizotinibKinase InhibitorALK, ROS1, MET
28CyclophosphamideAlkylating AgentDNA (Cross-linking)
29CyclosporineImmunosuppressantCalcineurin
30CytarabineAntimetaboliteDNA Polymerase (via Ara-C)
31DabrafenibKinase InhibitorBRAF (V600E/K mutation)
32DacomitinibKinase InhibitorEGFR (ErbB1), HER2, ErbB4
33DaraxonrasibRAS inhibitorActive RAS proteins
34DasatinibKinase InhibitorBCR-ABL, SRC Family, c-KIT
35DaunorubicinAntitumor AntibioticDNA (Intercalation) / Topoisomerase II
36DecitabineAntimetabolite (Epigenetic)DNMT (DNA Methyltransferase)
37DefactinibInvestigational InhibitorFAK (Focal Adhesion Kinase)
38DeferasiroxIron ChelatorIron (Fe3+)
39DexamethasoneCorticosteroidGlucocorticoid Receptor
40DocetaxelAnti-Microtubule AgentMicrotubules (Stabilization)
41DoxorubicinAntitumor AntibioticDNA (Intercalation) / Topoisomerase II
42DuvelisibKinase InhibitorPI3K (Delta, Gamma isoforms)
43EnasidenibMetabolic InhibitorIDH2 (Isocitrate Dehydrogenase 2)
44EncorafenibKinase InhibitorBRAF (V600E)
45EntrectinibKinase InhibitorNTRK, ROS1, ALK
46EpirubicinAntitumor AntibioticDNA (Intercalation) / Topoisomerase II
47EribulinAnti-Microtubule AgentMicrotubules (Destabilization)
48ErlotinibKinase InhibitorEGFR (Tyrosine Kinase)
49EtoposideTopoisomerase InhibitorTopoisomerase II
50EverolimusKinase Inhibitor (mTOR)mTORC1
51FludarabineAntimetaboliteDNA Polymerase / Ribonucleotide Reductase
52FruquintinibKinase InhibitorVEGFR 1, 2, 3
53GefitinibKinase InhibitorEGFR (Tyrosine Kinase)
54GemcitabineAntimetaboliteDNA Chain Elongation / Ribonucleotide Reductase
55GilteritinibKinase InhibitorFLT3, AXL
56IdarubicinAntitumor AntibioticDNA (Intercalation) / Topoisomerase II
57IfosfamideAlkylating AgentDNA (Cross-linking)
58ImatinibKinase InhibitorBCR-ABL, KIT, PDGFR
59InobrodibInvestigational Epigenetic Modifierp300 / CBP (Histone Acetyltransferases)
60Irinotecan (SN-38)Topoisomerase InhibitorTopoisomerase I
61IvosidenibMetabolic InhibitorIDH1 (Isocitrate Dehydrogenase 1)
62IxazomibProteasome Inhibitor20S Proteasome (Beta-5 subunit)
63L-AsparaginaseEnzymeAsparagine (Amino Acid Depletion)
64LapatinibKinase InhibitorEGFR, HER2
65LazertinibKinase InhibitorEGFR (Mutation specific)
66LenalidomideImmunomodulator (IMiD)Cereblon (E3 Ubiquitin Ligase)
67LenvatinibKinase InhibitorVEGFR, FGFR, PDGFR, RET, KIT
68LetrozoleHormonal TherapyAromatase (CYP19A1)
69MelphalanAlkylating AgentDNA (Cross-linking)
70MethotrexateAntimetaboliteDihydrofolate Reductase (DHFR)
71MidostaurinKinase InhibitorFLT3, KIT
72MirvetuximabAntibody-Drug ConjugateFolate Receptor Alpha (FRα)
73Mitomycin CAntitumor AntibioticDNA (Cross-linking/Alkylation)
74MitoxantroneAntitumor AntibioticTopoisomerase II / DNA Intercalation
75NilotinibKinase InhibitorBCR-ABL
76NiraparibPARP InhibitorPARP1, PARP2
77OlaparibPARP InhibitorPARP1, PARP2, PARP3
78OxaliplatinAlkylating AgentDNA (Cross-linking)
79PaclitaxelAnti-Microtubule AgentMicrotubules (Stabilization)
80PalbociclibKinase InhibitorCDK4, CDK6
81PanobinostatEpigenetic ModifierHistone Deacetylases (Pan-HDAC)
82PazopanibKinase InhibitorVEGFR, PDGFR, KIT
83PemetrexedAntimetaboliteDHFR, Thymidylate Synthase, GARFT
84PomalidomideImmunomodulator (IMiD)Cereblon (E3 Ubiquitin Ligase)
85PonatinibKinase InhibitorBCR-ABL (including T315I), VEGFR, FGFR
86ProcarbazineAlkylating AgentDNA / RNA / Protein Synthesis
87QuizartinibKinase InhibitorFLT3
88RegorafenibKinase InhibitorVEGFR, TIE2, KIT, RET, RAF
89RevumenibEpigenetic ModifierMenin (Menin-KMT2A Interaction)
90RipretinibKinase InhibitorKIT, PDGFRA (Switch Pocket)
91RomidepsinEpigenetic ModifierHistone Deacetylases (HDAC1, HDAC2)
92RuxolitinibKinase InhibitorJAK1, JAK2
93SelinexorNuclear Export InhibitorXPO1 (Exportin 1)
94SorafenibKinase InhibitorVEGFR, PDGFR, RAF
95SotorasibKinase InhibitorKRAS G12C
96SunitinibKinase InhibitorVEGFR, PDGFR, KIT, FLT3
97TamoxifenHormonal TherapyEstrogen Receptor (ER)
98TemozolomideAlkylating AgentDNA (O6-guanine methylation)
99ThalidomideImmunomodulator (IMiD)Cereblon (E3 Ubiquitin Ligase) / VEGF
100TipiracilAntimetaboliteThymidine Phosphorylase (Protects Trifluridine)
101TopotecanTopoisomerase InhibitorTopoisomerase I
102TrabectedinAlkylating AgentDNA Minor Groove
103TrametinibKinase InhibitorMEK1, MEK2
104TrifluridineAntimetaboliteDNA (Incorporation)
105Valproic AcidEpigenetic ModifierHistone Deacetylase (HDAC)
106VenetoclaxApoptosis InducerBCL-2
107VincristineAnti-Microtubule AgentMicrotubules (Inhibition of Polymerization)
108VinorelbineAnti-Microtubule AgentMicrotubules (Inhibition of Polymerization)
109ZanubrutinibKinase InhibitorBTK (Bruton's Tyrosine Kinase)

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